51827-14-6Relevant articles and documents
MALT1 INHIBITORS AND USES THEREOF
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Paragraph 00324; 00325; 00328, (2019/08/15)
Provided herein are compounds of Formula (I) and pharmaceutical compositions thereof, which may be useful as MALT1 inhibitors. Also provided are for the treatment of proliferative disorders (e.g., cancer (e.g., non-Hodgkin' s lymphoma, diffuse large B-cell lymphoma, MALT lymphoma), benign neoplasm, a disease associated with angiogenesis,an autoimmune disease, an inflammatory disease, an autoinflammatory disease) by administering a compound of Formula (I).
Expeditious amide-forming reactions using thiol esters
Kurosu, Michio
, p. 591 - 594 (2007/10/03)
The reaction of a 2-pyridylthiol ester with a dimethylaluminum amide leads to the rapid formation of the corresponding amide. The tolylthiol esters can be activated with silver trifluoroacetate and coupled even with poorly reactive amino compounds. (C) 20
Rapid, one-pot synthesis of urethane-protected tripeptides
Zhu, Yun-Fei,Fuller, William D.
, p. 807 - 810 (2007/10/02)
Urethane-protected tripeptides are synthesized in solution, without isolation of purification of intermediates, using urethane-protected N-carboxyanhydrides as coupling reagents and hydrogenation for removal of N-protection.
