Organic Letters
Letter
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(h) Zhang, T.; Qi, Z.; Zhang, X.; Wu, L.; Li, X. Chem. - Eur. J. 2014,
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functionalization process, the three-component assembly of
quinolines could be achieved.
ASSOCIATED CONTENT
* Supporting Information
■
S
The Supporting Information is available free of charge on the
Experimental procedures and full characterization for all
compounds
(11) Lenden, P.; Entwistle, D. A.; Willis, M. C. Angew. Chem., Int. Ed.
2011, 50, 10657.
AUTHOR INFORMATION
Corresponding Author
(12) Murphy, S. K.; Bruch, A.; Dong, V. M. Angew. Chem., Int. Ed.
2014, 53, 2455.
(13) Castaing, M.; Wason, S. L.; Estepa, B.; Hooper, J. F.; Willis, M.
C. Angew. Chem., Int. Ed. 2013, 52, 13280.
(14) Du, X.-W.; Stanley, L. M. Org. Lett. 2015, 17, 3276.
(15) (a) Chaplin, A. B.; Hooper, J. F.; Weller, A. S.; Willis, M. C. J.
Am. Chem. Soc. 2012, 134, 4885. (b) Pernik, I.; Hooper, J. F.; Chaplin,
A. B.; Weller, A. S.; Willis, M. C. ACS Catal. 2012, 2, 2779.
(16) Hooper, J. F.; Chaplin, A. B.; Gonzalez-Rodríguez, C.;
́
Thompson, A. L.; Weller, A. S.; Willis, M. C. J. Am. Chem. Soc.
2012, 134, 2906.
(17) Hooper, J. F.; Young, R. D.; Pernik, I.; Weller, A. S.; Willis, M.
C. Chem. Sci. 2013, 4, 1568.
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Heterocycles 2006, 68, 1675. (b) Okuma, K.; Seto, J.-I.; Nagahora, N.;
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Notes
The authors declare no competing financial interest.
ACKNOWLEDGMENTS
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We thank the EPSRC, and Eli Lilly and Company for support
of this study.
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