Development of the first and practical method for enantioselective synthesis of 10B-enriched p-borono-l-phenylalanine

DOI: 10.1016/j.tetlet.2008.05.108

Source and publish data:

Tetrahedron Letters p. 4977 - 4980 (2008)

Update date:2022-07-30

Topics:

Authors:

Hattori, Yoshihide

Asano, Tomoyuki

Kirihata, Mitsunori

Yamaguchi, Yoshihiro

Wakamiya, Tateaki

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Article abstract of DOI:10.1016/j.tetlet.2008.05.108

At present p-(¹⁰B)borono-l-phenylalanine (l-¹⁰Bpa) is used clinically as an excellent ¹⁰B carrier for BNCT; however, its enantioselective synthesis has not been reported yet. The present Letter describes the first and prac

Full text of DOI:10.1016/j.tetlet.2008.05.108

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Product name:N^α-benzyloxycarbonyl-p-[2,3-dihydro-1H-naphtho[1,8-de]-1,3-diaza-2-(10B)borinyl]-L-phenylalanine methyl ester

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