Bioorganic and Medicinal Chemistry (2017)
Update date:2022-08-04
Topics:
Ogiyama, Tomoko
Yamaguchi, Mitsuhiro
Kurikawa, Nobuya
Honzumi, Shoko
Terayama, Koji
Nagaoka, Nobumi
Yamamoto, Yuka
Kimura, Takako
Sugiyama, Daisuke
Inoue, Shin-ichi
HSL inhibition is a promising approach to the treatment of dyslipidemia. As a result of re-optimization of lead compound 2, we identified novel compound 25a exhibiting potent inhibitory activity against HSL enzyme and cell with high selectivity for cholin
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