European Journal of Medicinal Chemistry p. 179 - 186 (1987)
Update date:2022-08-05
Topics:
Lachance, Bernard
Salvador, Romano L.
Simon, David Z.
Ten acetylenic esters, amides and Nδ-alkynyl derivatives of serine, 2,3-diaminopropanoic acid and glutamine were prepared as potential phosphoribosyl pyrophosphate amidotransferase (EC 2.4.2.14) inhibitors as well as anti-tumor agents against e
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