Studies on Organophosphorus Compounds; Part XX. A Facile Synthesis of α-Amino-Substituted Benzylphosphonic and -phosphinic Acids by Use of Thiophosphoramide

DOI: 10.1055/s-1986-31790

Source and publish data:

Synthesis p. 821 - 825 (1986)

Update date:2022-07-30

Topics: Synthesis Organic compounds Organophosphorus compounds Functional Groups Facile Synthesis

Authors:

Yuan, Chengye

Qi, Youmao

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Article abstract of DOI:10.1055/s-1986-31790

A facile method for the preparation of α-amino-substituted benzylphosphonic and -phosphinic acids is reported.It consists of the reaction of O,O-diethyl or O-ethyl O-phenyl phosphoroamidothioate (1) with a substituted benzaldehyde (2) and a phosphorous or

Full text of DOI:10.1055/s-1986-31790

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