Investigation of the structural parameters involved in the μ and δ opioid receptor discrimination of linear enkephalin-related peptides

DOI: 10.1021/jm00397a019

Source and publish data:

Journal of Medicinal Chemistry p. 374 - 383 (1988)

Update date:2022-09-26

Topics: Experimental Design

Authors:

Gacel Gacel

Zajac Zajac

Delay-Goyet

Dauge Dauge

Roques Roques

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Article abstract of DOI:10.1021/jm00397a019

The previous rules proposed for selective recognition of μ and δ opioid receptors by modified enkephalins were investigated through an extensive structure-activity study. Thus, modifications of the sequence of TRIMU 4 (Tyr-D-Ala-Gly-NHCH(CH₃)CH

Full text of DOI:10.1021/jm00397a019

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