Investigation of the structural parameters involved in the μ and δ opioid receptor discrimination of linear enkephalin-related peptides

DOI: 10.1021/jm00397a019

Source and publish data:

Journal of Medicinal Chemistry p. 374 - 383 (1988)

Update date:2022-09-26

Topics: Experimental Design

Authors:

Gacel Gacel

Zajac Zajac

Delay-Goyet

Dauge Dauge

Roques Roques

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1021/jm00397a019

The previous rules proposed for selective recognition of μ and δ opioid receptors by modified enkephalins were investigated through an extensive structure-activity study. Thus, modifications of the sequence of TRIMU 4 (Tyr-D-Ala-Gly-NHCH(CH₃)CH

Full text of DOI:10.1021/jm00397a019

Products guided by the article

Product name:L-Leucine, N-[N-[N-[(1,1-dimethylethoxy)carbonyl]glycyl]-L-phenylalanyl]-N-methyl-, phenylmethyl ester

Cas No:112575-05-0

R&D Labs maybe for 112575-05-0

Shandong Dayi Chemical Co., Ltd.

website:http://www.dayi.com.cn

Contact:+86- 535-7388728. 15306386031

Address:No 1 Danya west road, Laiyang City, Shandong province
Chengdu CSH Pharmaceutical Co.,ltd

Contact:+86-(28)-85321971

Address:Block B,New Hope Int. Tian Fu New District, Chengdu, Sichuan, China
JIANGXI ZHANGFENG CHEMICAL CO., LTD.

Contact:+86-0799-3413066

Address:Xiyuan village, Xiabu Town, Xiangdong District
Nanjing Fayekong Chemcial Co.,Ltd(expird)

Contact:86-25-58813444

Address:Rm 1503, Unit 1, Building 5, Zijinnanyuan, Nanjing, Jiangsu, China
Xuzhou Tianrun Chemical Co.,Ltd

website:http://www.tianrunchem.cn

Contact:86-516-83832636

Address:fuxing road

Relevant to this article

Dansyl-anthracene dyads for ratiometric fluorescence recognition of Cu ²⁺

Doi:10.1039/c0dt01016b
(2011)
Synthesis of μ-Carbene and μ-Carbyne Complexes of Rhodium and Cobalt from Substituted Diazirines. Crystal Structures of 5-C5Me5)2(CO)2<μ-C(C6H4F-4)(OMe)>> and 5-C5Me5)2(μ-CO)(μ-C6H4Me-4)>

Doi:10.1039/DT9910001417
(1991)
Synthesis and modifications of a small library of 1,4-benzodiazepin-3-ones toward potential inhibitors of the collagen-von Willebrand Factor interaction

Doi:10.1016/j.tet.2009.03.095
(2009)
Assembly of Diversely Substituted Quinolines via Aerobic Oxidative Aromatization from Simple Alcohols and Anilines

Doi:10.1021/acs.joc.6b03064
(2017)
Synthesis and α₂-Adrenoceptor Antagonist Activity of Some Disulfonamidobenzoquinolizines

Doi:10.1021/jm00121a033
(1989)
Novel tricyclic pyrazolopyrimidines as potent and selective GPR119 agonists

Doi:10.1016/j.bmcl.2014.10.010
(2014)

Article Doi