
Journal of Medicinal Chemistry p. 1968 - 1971 (1988)
Update date:2022-09-26
Topics:
Glennon, Richard A.
Naiman, Noreen A.
Lyon, Robert A.
Titeler, Milt
Although simple arylpiperazines are commonly considered to be moderately selective for 5-HT1B serotonin binding sites, N4-substitution of such compounds can enhance their affinity for 5-HT1A sites and/or decrease their affinity for 5
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