Diastereo- and Enantio-selective Synthesis of Dihydro- and Tetrahydro-pyrimidines. A New Strategy for the Asymmetric Synthesis of β-Amino Ketones and γ-Amino Alcohols

DOI: 10.1039/C3988000410b

Source and publish data:

Journal of the Chemical Society. Chemical communications p. 410 - 412 (1988)

Update date:2022-08-04

Topics:

Authors:

Barluenga, Jose

Olano, Bernardo

Fustero, Santos

Foces-Foces, M. de la Concepcion

Cano, Felix Hernandez

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1039/C3988000410b

Chiral 1,2-dihydro- (3) and 1,2,3,6-tetrahydro-pyrimidines (4) have been synthesized by reaction of 3-aminoalk-2-enimines (1) with chiral aldehydes, the structure of (4) being comfirmed by an X-ray crystal structure determination of a reduction product; a

Full text of DOI:10.1039/C3988000410b

View Article Online / Journal Homepage / Table of Contents for this issue

View Article Online

Products guided by the article

Product name:(1R,2S)-2-((S)-1-Benzyloxy-ethyl)-5-methyl-1,6-diphenyl-4-p-tolyl-1,2-dihydro-pyrimidine

Cas No:117596-58-4

R&D Labs maybe for 117596-58-4

Cangzhou Senary Chemical Science-tech Co., Ltd

Contact:+86-317-3563899, 3563699

Address:168 Jinde Road, Cangzhou, Hebei, China
Evershine Chemical CO Ltd

Contact:+86-571-87010026

Address:202, Zhenhua Road,
Shanghai Yuking Water Soluble Material Tech Co., Ltd

Contact:86-21-68286299

Address:4F, 13B, No. 600, South Xinyuan Road 201306, Shanghai, China
Zhejiang Tianyu Pharmaceutical Co., Ltd.

Contact:+86-576-84177669, 89189665,89189688,84168770

Address:Jiangkou Development Zone, Huangyan, Taizhou City, Zhejiang
Beijing eternalchem Co,. Ltd

Contact:+86-10-59484199

Address:No.58-A1026 Liangguan Street

Relevant to this article

Synthesis and biological activity of some novel thieno[2,3-b]quinoline, quinolino[3′,2′-4,5] thieno[3,2-d]pyrimidine and pyrido[2′,3′:4,5] thieno[2,3-b]quinoline derivatives

Doi:10.1080/104265090970322
(2006)
Ru^II-catalyzed vinylative dearomatization of naphthols via a C(sp²)-H bond activation approach

Doi:10.1021/ja410060e
(2013)
Polyarylated thiazoles via a combined halogen dance - Cross-coupling strategy

Doi:10.1002/ejoc.200900092
(2009)
P-chirogenic benzo-fused phenoxaphosphane: Synthesis, resolution and study of the stereochemical properties of the corresponding palladium complexes

Doi:10.1002/ejic.200700887
(2008)
Doi:10.1038/135994a0
()
Nucleosides. 150. Synthesis and some biological properties of 5-monofluoromethyl, 5-difluoromethyl, and 5-trifluoromethyl derivatives of 2'-deoxyuridine and 2'-deoxy-2'-fluoro-β-D-arabinofuranosyluracil

Doi:10.1021/jm00403a026
(1988)

Article Doi