Diastereo- and Enantio-selective Synthesis of Dihydro- and Tetrahydro-pyrimidines. A New Strategy for the Asymmetric Synthesis of β-Amino Ketones and γ-Amino Alcohols

DOI: 10.1039/C3988000410b

Source and publish data:

Journal of the Chemical Society. Chemical communications p. 410 - 412 (1988)

Update date:2022-08-04

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Authors:

Barluenga, Jose

Olano, Bernardo

Fustero, Santos

Foces-Foces, M. de la Concepcion

Cano, Felix Hernandez

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Article abstract of DOI:10.1039/C3988000410b

Chiral 1,2-dihydro- (3) and 1,2,3,6-tetrahydro-pyrimidines (4) have been synthesized by reaction of 3-aminoalk-2-enimines (1) with chiral aldehydes, the structure of (4) being comfirmed by an X-ray crystal structure determination of a reduction product; a

Full text of DOI:10.1039/C3988000410b

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