Bioorganic and Medicinal Chemistry Letters p. 4380 - 4384 (2009)
Update date:2022-08-04
Topics:
Coon, Timothy
Moree, Wilna J.
Li, Binfeng
Yu, Jinghua
Zamani-Kord, Said
Malany, Siobhan
Santos, Mark A.
Hernandez, Lisa M.
Petroski, Robert E.
Sun, Aixia
Wen, Jenny
Sullivan, Sue
Haelewyn, Jason
Hedrick, Michael
Hoare, Samuel J.
Bradbury, Margaret J.
Crowe, Paul D.
Beaton, Graham
The benzimidazole core of the selective non-brain-penetrating H1-antihistamine mizolastine was used to identify a series of brain-penetrating H1-antihistamines for the potential treatment of insomnia. Using cassette PK studies, brain
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(2009)Doi:10.1002/chem.200900230
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(2009)Doi:10.1016/j.tetasy.2009.05.026
(2009)