Bioorganic and Medicinal Chemistry Letters p. 6064 - 6067 (2013)
Update date:2022-08-04
Topics:
Atobe, Masakazu
Naganuma, Kenji
Kawanishi, Masashi
Morimoto, Akifumi
Kasahara, Ken-Ichi
Ohashi, Shigeki
Suzuki, Hiroko
Hayashi, Takahiko
Miyoshi, Shiro
We describe a medicinal chemistry approach to generate a series of 2-(1H-pyrazol-1-yl)thiazole compounds that act as selective EP1 receptor antagonists. The obtained results suggest that compound 12 provides the best EP1 receptor ant
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