Organic Letters
Letter
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̌
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(13) For the single crystal information of 5f, see the Supporting
(14) For this novel Ag-catalyzed C−P bond formation reaction, we are
currently exploring its possible mechanism and will report it in due
course.
(15) For the single crystal information of 9, see the Supporting
(16) Patnaik, S.; Marugan, J. J.; Liu, K.; Zheng, W.; Southall, N.;
Dehdashti, S. J.; Thorsell, A.; Heilig, M.; Bell, L.; Zook, M.; Eskay, B.;
Brimacombe, K. R.; Austin, C. P. J. Med. Chem. 2013, 56, 9045.
(17) Possibly, the chemical stability of N-(2-pyridyl)imino chloride F is
poorer than that of N-phenylimino chloride 12, so we did not obtain the
corresponding spectral data about intermediate F.
D
Org. Lett. XXXX, XXX, XXX−XXX