Conformationally restricted P1-P1' transition analogues. Synthesis of 1(R), 3(R) [1(S), 2(S)] and 1(S), 3(S) [1(S),2(S)] 3-[3-cyclohexyl-2-[(BOC)amino]-1-hydroxypropyl]-2,2-dimethylcycloprop ane carboxylic acids

Article abstract of DOI:10.1016/S0040-4039(00)94403-4

A concise synthesis and determination of absolute stereochemistry of two novel diastereomeric cyclopropyl containing transition state mimics is described.