
Journal of Medicinal Chemistry p. 2045 - 2051 (1990)
Update date:2022-09-26
Topics:
McNamara
Berman
Fry
Werbel
The synthesis and biological activity of two series of nonclassical thymidylate synthase (TS) inhibitors are described. The first is a series of 10-propargyl-5.8-dideazafolic acid derivatives (10a-j) and the second is a series of the analogous 2-desamino
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Doi:10.1021/jm100582w
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(1989)