A novel chiral oxazolidine organocatalyst for the synthesis of an oseltamivir intermediate using a highly enantioselective Diels-Alder reaction of 1,2-dihydropyridine

DOI: 10.1039/c0cc00110d

Source and publish data:

Chemical Communications p. 4827 - 4829 (2010)

Update date:2022-09-26

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Authors:

Nakano, Hiroto

Osone, Kenichi

Takeshita, Mitsuhiro

Kwon, Eunsang

Seki, Chigusa

Matsuyama, Haruo

Takano, Nobuhiro

Kohari, Yoshihito

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Article abstract of DOI:10.1039/c0cc00110d

Enantioselective Diels-Alder reactions of 1,2-dihydropyridines with acroleins using a novel chiral oxazolidine organocatalyst afforded chiral isoquinuclidines that is an efficient synthetic intermediate of oseltamivir, with fairly good chemical yield and

Full text of DOI:10.1039/c0cc00110d

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Product name:(2S,4S)-4-tert-butyl-2,5,5-triphenyl-oxazolidine trifluoroacetate

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