Reactions of Benzotriazole with Formaldehyde and Aliphatic Primary Amines: Selective Formation of 1:1:1, of 2:2:1, and of 2:3:2 Adducts and a Study of their Reactions with Nucleophiles

DOI: 10.1039/P19900000541

Source and publish data:

Journal of the Chemical Society. Perkin transactions I p. 541 - 547 (1990)

Update date:2022-07-30

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Authors:

Katritzky, Alan R.

Pilarski, Boguslaw

Urogdi, Laszlo

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Article abstract of DOI:10.1039/P19900000541

Benzotriazole (BtH) reacts easily with aliphatic primary amines and formaldehyde in aqueous media to give one or more of three types of product: (i) (BtCCH2)2NR (5), (ii) (BtCH2NR)2CH2 (6), and/or (iii) BtCH2NHR (7).The product formed depends on the molar

Full text of DOI:10.1039/P19900000541

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