Design of Potent and Selective Linear Antagonists of Vasopressor (V1-Receptor) Responses to Vasopressin

DOI: 10.1021/jm00173a027

Source and publish data:

Journal of Medicinal Chemistry p. 3079 - 3086 (1990)

Update date:2022-07-30

Topics:

Authors:

Manning, Maurice

Stoev, Stoytcho

Kolodziejczyk, Aleksander

Klis, Wieslaw A.

Kruszynski, Marian

et al. et al.

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Article abstract of DOI:10.1021/jm00173a027

We report the solid-phase synthesis of 21 linear analogues of A and D, two nonselective antagonists of the vasopressor (V₁) and antidiuretic (V₂) responses to arginine vasopressin (AVP).A is Aaa-D-Tyr(Et)-Phe-Val-Asn-Abu-Pro-Arg-Arg-

Full text of DOI:10.1021/jm00173a027

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