Design of Potent and Selective Linear Antagonists of Vasopressor (V1-Receptor) Responses to Vasopressin

DOI: 10.1021/jm00173a027

Source and publish data:

Journal of Medicinal Chemistry p. 3079 - 3086 (1990)

Update date:2022-07-30

Topics:

Authors:

Manning, Maurice

Stoev, Stoytcho

Kolodziejczyk, Aleksander

Klis, Wieslaw A.

Kruszynski, Marian

et al. et al.

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1021/jm00173a027

We report the solid-phase synthesis of 21 linear analogues of A and D, two nonselective antagonists of the vasopressor (V₁) and antidiuretic (V₂) responses to arginine vasopressin (AVP).A is Aaa-D-Tyr(Et)-Phe-Val-Asn-Abu-Pro-Arg-Arg-

Full text of DOI:10.1021/jm00173a027

Products guided by the article

Product name:1-adamantylacetyl-D-Tyr(Et)-Phe-Val-Asn-Arg(Tos)-Pro-Arg(Tos)-Arg(Tos)-NH₂

Cas No:129520-72-5

R&D Labs maybe for 129520-72-5

Weifang Yukai Chemical Co.,Ltd.

website:http://www.yukaichem.com/en.html

Contact:+86-536-8865336

Address:binhai economic development zone，262737 shangdong，china
SINO Industries Company Limited(expird)

Contact:86-29-85369724

Address:No.111, Jiefang Road, Xi’an, China
Wuhan Honor Bio-Pharm Co., Ltd

Contact:0086-027-88042901

Address:Suite 1420, No.9 Building, Wanda Plaza, No.209 Heping Avenue, Wuchang District, Wuhan City, Hubei Province, P.R.China
Jinan Jinguilin Chemical Co.,Ltd

Contact:+86-531-81188412

Address:3rd floor of Torch Building, Huanyuan Rd, City of Jinan
Wuxi Olite Chemical Co., Ltd.

Contact:86-510-82853889

Address:Rm.3732, No.18-2,Yonghe Rd.,Wuxi,Jiangsu,214023,China

Relevant to this article

New simple wittig-type cyclizations to flavones, 4-quinolones and indenones¹

Doi:10.1016/S0040-4020(01)81518-0
(1990)
Microwave-assisted aminocarbonylation of ynamides by using catalytic [Fe₃(CO)₁₂] at low pressures of carbon monoxide

Doi:10.1002/chem.201100447
(2011)
Rapid access to unusual solid-state luminescent merocyanines by a novel one-pot three-component synthesis

Doi:10.1021/ol200655s
(2011)
PEGPHOT: A new well-defined molecular weight polyether-substituted triphenylphosphite and its application in biphasic hydroformylation

Doi:10.1007/s10562-011-0603-5
(2011)
Mechanism of Dicyanoanthracene-Photosensitized Oxygenation of 1,1,2,2-Tetraarylcyclopropanes and 1,1,3,3-Tetraarylpropenes

Doi:10.1021/jo00311a011
(1990)
A new one-pot synthesis of dialkyl phosphonates from diazo compounds and dialkyl hydrogen phosphites

Doi:10.1055/s-1990-26924
(1990)

Article Doi