Enantioselective total synthesis of aperidine

DOI: 10.1021/ol200728w

Source and publish data:

Organic Letters p. 2789 - 2791 (2011)

Update date:2022-08-04

Topics:

Authors:

Wakimoto, Toshiyuki

Miyata, Kakeru

Ohuchi, Hitoshi

Asakawa, Tomohiro

Nukaya, Haruo

Suwa, Yoshihide

Kan, Toshiyuki

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Article abstract of DOI:10.1021/ol200728w

An efficient total synthesis of aperidine was accomplished using a Rh-catalyzed C-H insertion of a cis-dihydrobenzofuran ring. To circumvent the facile epimerization of the cis-dihydrobenzofuran ring, we designed and prepared the C-H insertion precursor d

Full text of DOI:10.1021/ol200728w

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Product name:(2R,3S)-2-(4-(benzyloxy)phenyl)-N-(4-((tert-butyldimethylsilyl)oxy)butyl)-5-((E)-3-((4-((tert-butyldimethylsilyl)oxy)butyl)amino)-3-oxoprop-1-en-1-yl)-2,3-dihydrobenzofuran-3-carboxamide

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