Journal of Medicinal Chemistry p. 978 - 984 (1991)
Update date:2022-09-26
Topics:
Thornton
Jones
Jackman
Flinn
O'Connor
Warner
Calvert
We report the synthesis of four new 4-thio-5,8-dideazafolic acid analogues and a 4-(methylthio) analogue structurally related to the thymidylate synthase (TS) inhibitor N10-propargyl-5,8-dideazafolic acid. Three N10-propargyl-4-thio-
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(1990)