
Chemical and Pharmaceutical Bulletin p. 1411 - 1414 (1992)
Update date:2022-08-04
Topics:
Mavel
Coudert
Albuisson
Duroux
Bastide
Couquelet
Tronche
Rubat
N-Acetic acid derivatives of 6-aryl-pyrazolo-triazin-4-ones were synthesized for evaluation as new aldose reductase inhibitors. The intrinsic activity of each compound was assessed by measuring the inhibition of enzymatic activity in an isolated pig lens
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