2-Phenyl-3H-imidazopyridine-3-acetamides as Non-Benzodiazepine Anticonvulsants and Anxiolytics

DOI: 10.1021/jm00114a007

Source and publish data:

Journal of Medicinal Chemistry p. 2993 - 3006 (1991)

Update date:2022-08-05

Topics:

Authors:

Tomczuk, Bruce E.

Taylor, C. R

Moses, L. Meredith

Sutherland, Deborah B.

Lo, Young S.

et al. et al.

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Article abstract of DOI:10.1021/jm00114a007

A series of 2-phenyl-3H-imidazo<4,5-b>pyridine-3-acetamides were designed and synthesized as non-benzodiazepine anxiolytics based on a molecular disconnection of a typical 1,4-benzodiazepine (BZD).A number of these compounds showed submicromolar potency i

Full text of DOI:10.1021/jm00114a007

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