Conversion of avermectin B1 to 19-epi-avermectin B1

DOI: 10.1016/0040-4039(91)85068-G

Source and publish data:

Tetrahedron Letters p. 2723 - 2726 (1991)

Update date:2022-08-03

Topics:

Authors:

Blizzard

Bostrom Bostrom

Margiatto

Mrozik Mrozik

Fisher Fisher

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Article abstract of DOI:10.1016/0040-4039(91)85068-G

Avermectin B₁ (1) has been converted to 19-epi-avermectin B₁ (2) in six steps. Analog 2 retains some bioactivity but is substantially less bioactive than 1.

Full text of DOI:10.1016/0040-4039(91)85068-G

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