ACS Chemical Neuroscience p. 811 - 822 (2016)
Update date:2022-08-04
Topics:
Onajole, Oluseye K.
Vallerini, Gian Paolo
Eaton, J. Brek
Lukas, Ronald J.
Brunner, Dani
Caldarone, Barbara J.
Kozikowski, Alan P.
We report the synthesis and biological characterization of novel derivatives of 3-[(1-methyl-2(S)-pyrrolidinyl)methoxy]-5-cyclopropylpyridine (4a-f and 5) as potent and highly selective α4β2-nicotinic acetylcholine receptor (nAChR) full or partial agonist
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Doi:10.1021/ja00021a025
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