Chemical and Pharmaceutical Bulletin p. 2546 - 2555 (1994)
Update date:2022-08-05
Topics:
Kato
Ito
Nishino
Yamakuni
Takasugi
A series of pyrido[1,2-a]indol-6(7H)-ones was prepared and evaluated for 5-HT3 receptor antagonist activity. The structural requirements for the 5-HT3 receptor antagonist have been defined as an aromatic moiety, a basic nitrogen, and
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