Benzazepinone Calcium Channel Blockers. 3. Synthesis and Structure-Activity Studies of 3-Alkylbenzazepinones

DOI: 10.1021/jm00082a019

Source and publish data:

Journal of Medicinal Chemistry p. 773 - 780 (1992)

Update date:2022-07-29

Topics:

Authors:

Das, Jagabandhu

Floyd, David M.

Kimball, S. David

Duff, Keith J.

Vu, Truc Chi

et al. et al.

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Article abstract of DOI:10.1021/jm00082a019

As part of a program aimed at identifying novel analogues of diltiazem, we developed several synthetic routes for 3-alkylbenzazepinones, both in racemic and nonracemic form.Structure-activity relationship studies in this series have led to identification

Full text of DOI:10.1021/jm00082a019

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