Stereospecificity of amino acid side chains in deltorphin defines binding to opioid receptors

DOI: 10.1021/jm00085a009

Source and publish data:

Journal of Medicinal Chemistry p. 1222 - 1227 (1992)

Update date:2022-08-04

Topics:

Authors:

Lazarus Lazarus

Salvadori

Balboni Balboni

Tomatis Tomatis

Wilson Wilson

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Article abstract of DOI:10.1021/jm00085a009

A series of individual D-amino acid replacement analogues of deltorphin A, several of which were in combination with a His⁴ deletion, were used to probe alterations of side-chain orientation on peptide binding parameters with rat brain opioid r

Full text of DOI:10.1021/jm00085a009

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Product name:(D-Tyr¹,des-His⁴ )deltorphin A

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