Development of selective inhibitors against plasma kallikrein

DOI: 10.1248/cpb.39.2930

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 2930 - 2936 (1991)

Update date:2022-07-29

Topics:

Authors:

Teno Teno

Wanaka Wanaka

Okada Okada

Tsuda Tsuda

Okamoto Okamoto

Hijikata-Okunomiya

Naito Naito

Okamoto Okamoto

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1248/cpb.39.2930

Specific plasma kallikrein inhibitors were designed and synthesized and their structure-activity relationship was studied. trans-4-Aminomethylcyclohexanecarbonyl(Tra)-lysyl-4-ethoxycarbonylanili de inhibited plasma kallikrein and plasmin with 1C_{50
View More}

Full text of DOI:10.1248/cpb.39.2930

NII-Electronic Library Service

Products guided by the article

Product name:Benzoic acid, 4-[[5-[[imino(nitroamino)methyl]amino]-1-oxo-2-[[(phenylmethoxy)carbon yl]amino]pentyl]amino]-, 2-methylpropyl ester, (S)-

Cas No:140135-26-8

R&D Labs maybe for 140135-26-8

HENAN NEW BLUE CHEMICAL CO.,LTD

website:http://www.newbluechem.com

Contact:86-371-55170693/55170694

Address:Zhengzhou International Trade New Territory,Jinshui District,Zhengzhou ,China
Chengdu NoVi Biotechnology Co., Ltd.(expird)

Contact:13551243286/028-81458053

Address:NO.168-1-224 JULONG ROAD WUHOU DISTRICT, CHENGDU CITY,SICHUAN PROVINCE
Phantom-pharma

Contact:

Address:
Huangshan Violet Biological Technology Co., Ltd

Contact:+86-559-2335676

Address:16-201 JinShanYuan,JiangNan New City,TunXi District,HuangShan City,AnHui Province,China
Jiangxi Hessence Chemicals Co., Ltd.

Contact:+86 796 3511924

Address:Chengxi Industrial Park, Jishui County, Jiangxi Province 331600 China.

Relevant to this article

Application of ruthenium complexes of triazole-containing tridentate ligands to asymmetric transfer hydrogenation of ketones

Doi:10.1021/ol302354z
(2012)
Zn²⁺-selective fluorescent turn-on chemosensor based on terpyridine-substituted siloles

Doi:10.1016/j.dyepig.2012.04.007
(2012)
Fluorogenic detection of hydrogen sulfide via reductive unmasking of o-azidomethylbenzoyl-coumarin conjugate

Doi:10.1039/c2cc34682f
(2012)
Studies of asymmetric styrene cyclopropanation with a rhodium(II) metallopeptide catalyst developed with a high-throughput screen

Doi:10.1002/chir.22144
(2013)
The Discovery of a Potent, Selective, and Peripherally Restricted Pan-Trk Inhibitor (PF-06273340) for the Treatment of Pain

Doi:10.1021/acs.jmedchem.6b00850
(2016)
Sensitive near-infrared fluorescent probes for thiols based on Se-N bond cleavage: Imaging in living cells and tissues

Doi:10.1002/chem.201200671
(2012)

Article Doi