Structure-activity studies of a novel bicyclic oxytocin antagonist

DOI: 10.1021/jm00087a009

Source and publish data:

Journal of Medicinal Chemistry p. 1558 - 1563 (1992)

Update date:2022-08-05

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Authors:

Smith Smith

Slaninova

Hruby Hruby

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Article abstract of DOI:10.1021/jm00087a009

In this report, we describe structure-activity studies of the bicyclic oxytocin antagonist [Mpa¹,cyclo(Glu⁴,Lys⁸)]oxytocin. The monocyclic analogue [dPen¹,Glu⁴,Lys⁸]oxytocin was a weak oxyt

Full text of DOI:10.1021/jm00087a009

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