A concise asymmetric synthesis of the potent enkephalinase inihibitor kelatorphan

Article abstract of DOI:10.1080/00397919208020851

A concise asymmetric synthesis of the enkephalinase inhibitor Kelatorphan has been completed in seven steps from commercially available hydrocinnamyl chloride. The synthesis features as a key step an asymmetric C-C bond formation which utilizes Oppolzer b

Full text of DOI:10.1080/00397919208020851

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Synthetic Communications: An
International Journal for Rapid
Communication of Synthetic
Organic Chemistry
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A Concise Asymmetric
Synthesis of the Potent
Enkephalinase Inhibitor
Kelatorphan
Stevan W. Djuric a
a Gastrointestinal Diseases Research , Searle Skokie,
IL, 60077
Published online: 23 Sep 2006.
To cite this article: Stevan W. Djuric (1992) A Concise Asymmetric Synthesis of
the Potent Enkephalinase Inhibitor Kelatorphan, Synthetic Communications: An
International Journal for Rapid Communication of Synthetic Organic Chemistry, 22:6,
871-882, DOI: 10.1080/00397919208020851
To link to this article: http://dx.doi.org/10.1080/00397919208020851
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