Journal of Medicinal Chemistry p. 3156 - 3169 (1992)
Update date:2022-08-04
Topics:
Labaudiniere, Richard
Hilboll, Gerd
Leon-Lomeli, Alicia
Lautenschlaeger, Hans-Heiner
Parnham, Michael
et al.
The synthesis and structure-activity profile of a new class of potent and specific LTA4 hydrolase inhibitors are described.Many compounds of this series of ω-<5-(ω-arylalkyl)-2-thienyl>- and ω-<4-(ω-arylalkyl)phenyl>alkanoic acids were found to
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