Tandem coupling of 5-bromo-3-iodo-1-tosylindole with trimethylarylstannanes and aryl boronic acids

Article abstract of DOI:10.1080/00397919208020495

Palladium(0)-catalyzed coupling of 5-bromo-3-iodo-1-tosylindole with trimethylarylstannanes afforded 3-aryl-5-bromo-1-tosylindoles which were then coupled with aryl boronic acids to give 3,5-diarylated indoles in moderate to excellent yields.

Full text of DOI:10.1080/00397919208020495

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Synthetic Communications: An
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Organic Chemistry
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Tandem Coupling of 5-Bromo-3-
iodo-1-tosylindole with
Trimethylarylstannanes and
Aryl Boronic Acids
Youhua Yang a & Arnold R. Martin a
a Department of Pharmaceutical Sciences , College
of Pharmacy University of Arizona , Tucson, AZ,
85721
Published online: 23 Sep 2006.
To cite this article: Youhua Yang & Arnold R. Martin (1992) Tandem Coupling of 5-
Bromo-3-iodo-1-tosylindole with Trimethylarylstannanes and Aryl Boronic Acids,
Synthetic Communications: An International Journal for Rapid Communication of
Synthetic Organic Chemistry, 22:12, 1757-1762, DOI: 10.1080/00397919208020495
To link to this article: http://dx.doi.org/10.1080/00397919208020495
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