Handy access to chiral N,N'-disubstituted 3-aminopyrrolidines

DOI: 10.1016/S0957-4166(00)82081-9

Source and publish data:

Tetrahedron Asymmetry p. 1239 - 1242 (1992)

Update date:2022-07-30

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Authors:

Maddaluno

Corruble

Leroux Leroux

Ple Ple

Duhamel Duhamel

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Article abstract of DOI:10.1016/S0957-4166(00)82081-9

A new and rapid synthesis of (S)-3-aminopyrrolidines Z is proposed from N-protected (S)-Asparagine. Basic cyclization of methyl N-Z-(S)-Asparaginate 1 followed by one-pot N-benzylation directly leads to (S)-aminosuccinimide 3 which, after cleavage of the

Full text of DOI:10.1016/S0957-4166(00)82081-9

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