
Journal of Fluorine Chemistry p. 31 - 38 (1993)
Update date:2022-07-30
Topics:
Jarman, Michael
Bisset, Graham, M. F.
Thornton, Timothy J.
A synthesis of a tetrafluoro derivative of the quinazoline antifolate 2-desamino-2-methyl-N10-propargyl-5,8-dideazafolic acid is described. 2-Desamino-2-methyl-N10-propargyl-2',3',5',6'-tetrafluoro-5,8-dideazafolic acid (1) has been
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