Journal of Pharmacy and Pharmacology p. 63 - 66 (1993)
Update date:2022-08-03
Topics:
Zhang
Caldirola
Timmerman
Calcium channel affinity of terfenadine and its optical isomers was determined by the displacement of [3H]nitrendipine on rat cerebral cortex membranes. Terfenadine showed a pK(d) of 6.36 ± 0.03 whereas its R(+)-isomer (VUF4567) had a pK(d) val
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