Kynostatin (KNI)-227 and -272, highly potent anti-HIV agents: Conformationally constrained tripeptide inhibitors of HIV protease containing allophenylnorstatine

DOI: 10.1248/cpb.40.2251

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 2251 - 2253 (1992)

Update date:2022-07-29

Topics:

Authors:

Mimoto Mimoto

Imai Imai

Kisanuki

Enomoto Enomoto

Hattori Hattori

Akaji Akaji

Kiso Kiso

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Article abstract of DOI:10.1248/cpb.40.2251

Selective and potent HIV protease inhibitors containing allophenylnorstatine [Apns; (2S,3S)-3-amino-2-hydroxy-4-phenylbutyric acid] as a transition-state mimic were designed and synthesized. Among them, conformationally constrained tripeptide derivatives,

Full text of DOI:10.1248/cpb.40.2251

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