
Journal of Medicinal Chemistry p. 2300 - 2310 (1993)
Update date:2022-09-26
Topics:
Ghosh, Arun K.
Thompson, Wayne J.
Holloway, M. Katharine
McKee, Sean P.
Duong, Tien T.
et al.
A series of protease inhibitors bearing constrained unnaturel amino acids at the P2-position and novel heterocycles at the P3-position of compound 1 (Ro 31-8959) were synthesized, and their in vitro enzyme inhibitory and antiviral ac
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