
Tetrahedron Letters p. 977 - 980 (1994)
Update date:2022-08-05
Topics:
Dodd, Dharmpal S.
Kozikowski, Alan P.
An efficient method for the direct conversion of alcohols to guanidines is presented. A variety of alcohols react with 1 and 2 under Mitsunobu conditions to give the corresponding guanidines in high yield.
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