Amide bond formation via pentafluorothiophenyl active esters

DOI: 10.1016/S0040-4039(00)76989-9

Source and publish data:

Tetrahedron Letters p. 4865 - 4868 (1994)

Update date:2022-09-26

Topics:

Authors:

Davis, Anthony P.

Walsh, John J.

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Article abstract of DOI:10.1016/S0040-4039(00)76989-9

A number of pentafluorothiophenyl (PFTP) esters were shown to be useful acyl donors for amide bond formation, being non-polar, stable to chromatography and extended storage, but sufficiently active for use with relatively unreactive acyl groups. In partic

Full text of DOI:10.1016/S0040-4039(00)76989-9

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