A convergent synthesis of novel conformationally restricted HIV-1 protease inhibitors

DOI: 10.1016/S0040-4039(00)77051-1

Source and publish data:

Tetrahedron Letters p. 5153 - 5156 (1994)

Update date:2022-07-30

Topics:

Authors:

Kim, B. Moon

Guare, James P.

Hanifin, Colleen M.

Arford-Bickerstaff, Deborah J.

Vacca, Joseph P.

Ball, Richard G.

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Article abstract of DOI:10.1016/S0040-4039(00)77051-1

Conformationally restricted HIV-1 protease inhibitors containing the transition state hydroxyl group in pyrrolidine or piperidine ring systems were synthesized stereoselectively utilizing the inherent stereochemistry of an amino acid derivative. A converg

Full text of DOI:10.1016/S0040-4039(00)77051-1

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