
Tetrahedron Letters p. 5153 - 5156 (1994)
Update date:2022-07-30
Topics:
Kim, B. Moon
Guare, James P.
Hanifin, Colleen M.
Arford-Bickerstaff, Deborah J.
Vacca, Joseph P.
Ball, Richard G.
Conformationally restricted HIV-1 protease inhibitors containing the transition state hydroxyl group in pyrrolidine or piperidine ring systems were synthesized stereoselectively utilizing the inherent stereochemistry of an amino acid derivative. A converg
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(1994)Doi:10.1002/anie.201309521
(2014)Doi:10.1039/c7cc01606a
(2017)Doi:10.1039/c4cc00839a
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