(+)-cis-N-(Para-, meta-, and ortho-substituted benzyl)-N-normetazocines: Synthesis and binding affinity at the [3H]-(+)-pentazocine-labeled (σ1) site and quantitative structure-affinity relationship studies

DOI: 10.1021/jm00003a019

Source and publish data:

Journal of Medicinal Chemistry p. 565 - 569 (1995)

Update date:2022-08-03

Topics:

Authors:

Mascarella

Bai Bai

Williams

Sine Sine

Bowen Bowen

Carroll Carroll

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Article abstract of DOI:10.1021/jm00003a019

σ1 receptor ligands have potential pharmacological significance as antipsychotic drugs, as tools in the study of drug-induced motor function disorders, and as radiopharmaceutical imaging agents for the noninvasive imaging of malignant tumors in human subj

Full text of DOI:10.1021/jm00003a019

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