Synthesis of Functionalized Furopyridines via the Pd-catalyzed Coupling of Acetylenes to Iodopyridones. Preparation of a Key Intermediate to a New HIV Protease Inhibitor L-754,394.

DOI: 10.1016/S0040-4039(00)78541-8

Source and publish data:

Tetrahedron Letters p. 9355 - 9358 (1994)

Update date:2022-09-26

Topics:

Authors:

Houpis, Ioannis N.

Choi, W. B.

Reider, P. J.

Molina, Audrey

Churchill, Hywyn

et al. et al.

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Article abstract of DOI:10.1016/S0040-4039(00)78541-8

The synthesis of 1 was accomplished in 55percent overall yield via the Pd-catalyzed coupling of 3 and 4 followed by Cu-catalyzed cyclization of the resulting intermediate 2.

Full text of DOI:10.1016/S0040-4039(00)78541-8

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Product name:Furo[2,3-b]pyridine-5-carboxylic acid, ethyl ester

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