Chemical Biology and Drug Design p. 724 - 729 (2016)
Update date:2022-08-04
Topics:
Cosimelli, Barbara
Greco, Giovanni
Laneri, Sonia
Novellino, Ettore
Sacchi, Antonia
Trincavelli, Maria Letizia
Giacomelli, Chiara
Taliani, Sabrina
Da Settimo, Federico
Martini, Claudia
Three 4-amino-6-alkyloxy-2-alkylthiopyrimidine derivatives (4–6) were investigated as potential non-nucleoside agonists at human adenosine receptors (ARs). When tested in competition binding experiments, these compounds exhibited low micromolar affinity (
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