
Journal of Medicinal Chemistry p. 2145 - 2151 (1995)
Update date:2022-08-06
Topics:
Maruenda
Johnson
A variety of N1-substituted pyrimido[5,4-f]benzo[1,4]thiazepines, 5, designed as conformationally constrained analogs of 1-[(2- hydroxyethoxy)methyl]-6-(phenylthio)thymine HEPT (1), were synthesized and evaluated for their inhibition of human immunodefici
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