Molecules 2015, 20
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alternatively, ultrasonic activation of magnesium powder in DMF before addition of CFCl3 might be a
good option.
3.4. Characterization of the Products
All the products, 2a–e were identified by comparison of spectroscopic data (IR, 1H-NMR, 13C-NMR
and 19F-NMR) with the authentic samples as reported in [15,30,31]. The characteristic 1H-NMR values
are given below for reference:
2,2-Dichloro-2-fluoro-1-phenylethanol (2a). 1H-NMR (CDCl3): δ = 7.53 (m, 2H), 7.41 (m, 3H), 5.16 (d,
J = 8.4 Hz, 1H), 2.97 (br s, 1H, OH).
1
2,2-Dichloro-2-fluoro-1-(2-methylphenyl)ethanol (2b). H-NMR (CDCl3): δ = 7.66 (d, J = 6.9 Hz,
1H), 7.25 (m, 3H), 5.43 (d, J = 9.3 Hz, 1H), 2.60 (s, 3H), 3.05 (br s, 1H, OH).
1
2,2-Dichloro-2-fluoro-1-(2-chlorophenyl)ethanol (2c). H-NMR (CDCl3): δ = 7.75 (m, 1H), 7.36 (m,
3H), 5.77 (d, J = 9.3 Hz, 1H), 3.17 (br s, 1H, OH).
2,2-Dichloro-2-fluoro-1-(4-bromophenyl)ethanol (2d). 1H-NMR (CDCl3): δ = 7.53 (m, 2H), 7.40 (d,
J = 8.1 Hz, 2H), 5.11 (d, J = 7.5 Hz, 1H), 3.24 (br s, 1H, OH).
2,2-Dichloro-2-fluoro-1-(4-methoxyphenyl)ethanol (2e). 1H-NMR (CDCl3): δ = 7.45 (d, J = 8.4 Hz, 2H),
6.92 (d, J = 8.4 Hz, 2H), 5.10 (d, J = 8.7 Hz, 1H), 3.82 (s, 3H), 2.97 (br s, 1H, OH).
2,2-Dichloro-2-fluoro-1-(4-trifluoromethylphenyl)ethanol (2f). 1H-NMR (CDCl3): δ = 7.51 (m, 4H), 5.3
(d, J = 8.1 Hz, 1H), 3.1 (br s, 1H, OH).
1
2,2-Dichloro-2-fluoro-1-(4-fluorophenyl)ethanol (2g). H-NMR (CDCl3): δ = 7.75 (m, 2H), 7.36 (m,
2H), 5.8 (d, J = 9.1 Hz, 1H), 3.3 (br s, 1H, OH).
4. Conclusions
In conclusion, we present a cost-effective and facile method for the addition and modification of
aromatic aldehydes with CFCl3 under mild conditions. This method demonstrates a novel strategy for in
situ formation of a reactive dichlorofluoromethyl magnesium Grignard reagent and its importance in
synthesizing dichlorofluoromethyl aromatic alcohols. Unlike other previous methods, these reactions
can be performed under relatively mild conditions and can also be used in reactions with de-activated or
less electrophilic aromatic aldehyde substrates having electron donating substituents. However, the
yields obtained under these conditions are moderate. This is attributed to the in situ formation of
chlorofluorocarbene via a competing reaction pathway. Chlorofluorocarbene formation was verified via
isolation of the cyclopropane product (4), 1,1,2,2-tetramethylchlorofluorocyclopropane formed from the
reaction between tetramethylene (3) and chlrofluorocarbene. Based on previous reports [26–29], we
conclude that chlorofluorocarbene formation could have occurred with equal probability under the
employed reaction conditions, and further studies are needed to understand the kinetics and dependence
of the various factors/parameters.