Total synthesis of modified JSTX toxins: Reductive alkylation is a practical route to hexahydropyrimidine polyamine amides

DOI: 10.1016/0040-4039(95)01995-T

Source and publish data:

Tetrahedron Letters p. 9397 - 9400 (1995)

Update date:2022-08-03

Topics:

Authors:

Ashton, Mark R.

Moya, Eduardo

Blagbroug, Ian S.

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/0040-4039(95)01995-T

Reductive alkylation is a practical route for a total synthesis of regioisomers of spider toxin JSTX-3, a polyamine amide which is a selective glutamate receptor antagonist and may have potential as a neuroprotective agent. The strategy is based upon a re

Full text of DOI:10.1016/0040-4039(95)01995-T

Products guided by the article

Product name:(3-Benzyloxycarbonylamino-propyl)-(4-{benzyloxycarbonyl-[3-(5-{(S)-2-[2-(2,4-bis-benzyloxy-phenyl)-acetylamino]-3-carbamoyl-propionylamino}-pentylamino)-propyl]-amino}-butyl)-carbamic acid benzyl ester

Cas No:172992-26-6

R&D Labs maybe for 172992-26-6

Hangzhou Taiyan Trading Co., Ltd(expird)

Contact:+86-13777583958

Address:NO.63, Xingyi Street, Xihu District, Hangzhou, Zhejiang, China
Shanghai Send Pharmaceutical Technology Co., Ltd.

website:http://www.shsendpharma.com

Contact:021-58088081, +8613585868794

Address::Room A601, Building 1,NO. 800 Qingdai Road Pudong District Shanghai,China
Sichuan JieYao Co., Ltd.

Contact:+86-838-5655598

Address:Guanghan Nanfeng Industrial Zone
Chemieliva Pharmaceutical Co., Ltd.

website:http://www.chemieliva.com

Contact:+86-23-67770219

Address:99 Longhua Road, Yubei District, 401147, Chongqing, China Email: sales@chemieliva.com Tel:0086-23-67770219 Fax: 0086-23-67770220 Attn: Andy Huang
Nanjing Chemlin Chemical Co., Ltd.

website:http://www.echemlin.cn

Contact:+86-25-83697070

Address:Rm.902 Longyin Plaza, No. 217 Zhongshan Rd.(N) Nanjing 210009,China

Relevant to this article

A sulfated galactan with antioxidant capacity from the green variant of tetrasporic Gigartina skottsbergii (Gigartinales, Rhodophyta)

Doi:10.1016/j.carres.2011.11.014
(2012)
Complexation of o-(ethylphenylphosphino)(ethylthio)benzene towards nickel(II), palladium(II), and platinum(II) complexes

Doi:10.1080/10426509608029639
(1996)
Synthesis and evaluation of a polyamine phosphinate and phosphonamidate as transition-state analogue inhibitors of spermidine/spermine-N¹-acetyltransferase

Doi:10.1016/0968-0896(96)00072-7
(1996)
An improved method for the resolution of 1,1′-binaphthalene-2,2′-diol via a phosphite using (-)-menthol as a resolving agent

Doi:10.1080/10426500210215
(2002)
Study of pyrazidol metabolism

Doi:10.1007/BF02333964
(1996)
Eco-friendly H₂O₂ oxidation of 1,2-dihydroquinazoline-3-oxides to quinazoline-3-oxides

Doi:10.1080/00397911.2021.1934876
(2021)

Article Doi