Synthesis and evaluation of a polyamine phosphinate and phosphonamidate as transition-state analogue inhibitors of spermidine/spermine-N1-acetyltransferase

DOI: 10.1016/0968-0896(96)00072-7

Source and publish data:

Bioorganic and Medicinal Chemistry p. 825 - 836 (1996)

Update date:2022-08-03

Topics:

Authors:

Wu, Ronghui

Saab, Nada H.

Huang, Huatao

Wiest, Laurie

Pegg, Anthony E.

Casero Jr., Robert A.

Woster, Patrick M.

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/0968-0896(96)00072-7

Polyamine analogues such as bis(ethyl)norspermine and N¹-ethyl-N¹¹-[(cyclopropyl)methyl]-4,8-diazaundecane (CPENSpm) act as inhibitors of the enzyme spermidine/spermine-N¹-acetyltransferase (SSAT) in vitro and possess impr

Full text of DOI:10.1016/0968-0896(96)00072-7

Products guided by the article

Product name:1-{N-[benzyloxy(methyl)phosphinyl]amino}-3-[(N,N-dimethyl)amino]propane

Cas No:180523-55-1

R&D Labs maybe for 180523-55-1

SJZ Chenghui Chemical Co., Ltd.

Contact:86-311-87713916

Address:no.368 youyi north avenue
Jiaxing Carry Bio-Chem Technology Co.,Ltd

website:http://www.carrybiotech.com

Contact:0573-82788958

Address:Add.Fl 3th, Pharm Vally,Kaichuang Rd, Xiuzhou District, Jiaxing, Zhejiang,314031,China
SHUNYUANSHENG BIO-PHARMTECH CO., LTD

website:https://www.whsysbio.com

Contact:--

Address:Building 13, Liandong U Valley-Wuhan Economic Innovation Valley, No. 259, Xingsan Road, Shamao Street, Hannan District, Wuhan City, Hubei Province
Chengdu Baishixing Science and Technology Industry Co., Ltd.

website:http://www.cd-bsx.com

Contact:+86-28-88531548

Address:#217,North of Industry Road,Heshan Town,Pujiang County,Chengdu,Sichuan,China.
Nantong Auxin Electronic Technology Co., LTD

Contact:86-513-88760026

Address:NO.5-1, Aoxin Road, Haian Hi-tech Development Zone, Jiangsu Province, China

Relevant to this article

Synthesis of the D-3 series of phosphatidylinositol phosphates

Doi:10.1021/jo960602u
(1996)
Chemical approaches to bacterial vaccines. Synthesis of mycobacterial oligosaccharide-protein conjugates for use as serodiagnostics and immunogens

Doi:10.1016/0960-894X(96)00235-1
(1996)
Cleavage of titanium dimethylamides with methyl iodide

Doi:10.1021/om00019a057
(1994)
Studies on the standardization of crude drugs. XIX. The constituents of Picrasma ailanthoides. I. The structure of nigakinone

Doi:10.1248/yakushi1947.87.11_1371
(1967)
Unusual acetylation of 2-methyl-1-phenylsulfonylindole

Doi:10.1080/00397919608004636
(1996)
α-Diimine-Niobium Complex-Catalyzed Deoxychlorination of Benzyl Ethers with Silicon Tetrachloride

Doi:10.1021/acs.inorgchem.9b01784
(2019)

Article Doi