Synthesis and evaluation of a polyamine phosphinate and phosphonamidate as transition-state analogue inhibitors of spermidine/spermine-N1-acetyltransferase

DOI: 10.1016/0968-0896(96)00072-7

Source and publish data:

Bioorganic and Medicinal Chemistry p. 825 - 836 (1996)

Update date:2022-08-03

Topics:

Authors:

Wu, Ronghui

Saab, Nada H.

Huang, Huatao

Wiest, Laurie

Pegg, Anthony E.

Casero Jr., Robert A.

Woster, Patrick M.

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/0968-0896(96)00072-7

Polyamine analogues such as bis(ethyl)norspermine and N¹-ethyl-N¹¹-[(cyclopropyl)methyl]-4,8-diazaundecane (CPENSpm) act as inhibitors of the enzyme spermidine/spermine-N¹-acetyltransferase (SSAT) in vitro and possess impr

Full text of DOI:10.1016/0968-0896(96)00072-7

Products guided by the article

Product name:1-{N-[benzyloxy(methyl)phosphinyl]amino}-3-[(N,N-dimethyl)amino]propane

Cas No:180523-55-1

R&D Labs maybe for 180523-55-1

HEZE KINGVOLT CHEMICAL CO., LTD

Contact:86-573-82118911

Address:Juancheng Industry Park
Tianjin Boron PharmaTech Co.,Ltd.(expird)

Contact:86-022-59845187

Address:B9-401, Tianda Science Park,No.80,4th Avenue,TEDA,Tianjin, China
Acros Pharmatech Limited

website:http://www.acrospharmatech.com

Contact:+1-3234804688

Address:Flat/RM 1502,Easey Commercial building 253-261 Hennessy Road,Wanchai，HongKong
Jurong Huaheng Natural Biological Products Factory

website:http://www.risebiochem.com

Contact:+86-13921007726

Address:Chuncheng town,Jurong city,Jiangsu province,China
SJZ THLD IMP & EXP CO LTD

website:http://www.truewingroup.com

Contact:86-311-66699812

Address:NO.600 ZHONGSHAN EAST ROAD SHIJIAZHUANG

Relevant to this article

Synthesis of the D-3 series of phosphatidylinositol phosphates

Doi:10.1021/jo960602u
(1996)
Chemical approaches to bacterial vaccines. Synthesis of mycobacterial oligosaccharide-protein conjugates for use as serodiagnostics and immunogens

Doi:10.1016/0960-894X(96)00235-1
(1996)
Cleavage of titanium dimethylamides with methyl iodide

Doi:10.1021/om00019a057
(1994)
Studies on the standardization of crude drugs. XIX. The constituents of Picrasma ailanthoides. I. The structure of nigakinone

Doi:10.1248/yakushi1947.87.11_1371
(1967)
Unusual acetylation of 2-methyl-1-phenylsulfonylindole

Doi:10.1080/00397919608004636
(1996)
α-Diimine-Niobium Complex-Catalyzed Deoxychlorination of Benzyl Ethers with Silicon Tetrachloride

Doi:10.1021/acs.inorgchem.9b01784
(2019)

Article Doi