Synthesis and evaluation of a polyamine phosphinate and phosphonamidate as transition-state analogue inhibitors of spermidine/spermine-N1-acetyltransferase

DOI: 10.1016/0968-0896(96)00072-7

Source and publish data:

Bioorganic and Medicinal Chemistry p. 825 - 836 (1996)

Update date:2022-08-03

Topics:

Authors:

Wu, Ronghui

Saab, Nada H.

Huang, Huatao

Wiest, Laurie

Pegg, Anthony E.

Casero Jr., Robert A.

Woster, Patrick M.

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/0968-0896(96)00072-7

Polyamine analogues such as bis(ethyl)norspermine and N¹-ethyl-N¹¹-[(cyclopropyl)methyl]-4,8-diazaundecane (CPENSpm) act as inhibitors of the enzyme spermidine/spermine-N¹-acetyltransferase (SSAT) in vitro and possess impr

Full text of DOI:10.1016/0968-0896(96)00072-7

Products guided by the article

Product name:1-{N-[benzyloxy(methyl)phosphinyl]amino}-3-[(N,N-dimethyl)amino]propane

Cas No:180523-55-1

R&D Labs maybe for 180523-55-1

Hybio Pharmaceutica Co.,Ltd

website:http://www.hybio.com.cn

Contact:+86 755 26588093

Address:No.9 Linkong West Street, Hengdian Street, Huangpi District, Wuhan City, China.
Tianjin Ingenochem Technology Co.,Ltd

Contact:+86-22-23677060

Address:Hitech Green Industry Park K2-9-602, Nankai district
Hebei Think-Do Environment Co., Ltd

website:http://www.thinkdo-environment.com

Contact:0311-86510809-

Address:No 6, Shilian Middle Street, Circular Chemical Industry Park
Tianjin Ingenochem Technology Co.,Ltd

Contact:+86-22-23677060

Address:Hitech Green Industry Park K2-9-602, Nankai district
Jiangsu Cale New Material Co.ltd

Contact:+86-515-88334667/88203550

Address:Zhongshan 3rd Road, Coastal Chemical Industry Park, Yancheng, Jiangsu, China

Relevant to this article

Synthesis of the D-3 series of phosphatidylinositol phosphates

Doi:10.1021/jo960602u
(1996)
Chemical approaches to bacterial vaccines. Synthesis of mycobacterial oligosaccharide-protein conjugates for use as serodiagnostics and immunogens

Doi:10.1016/0960-894X(96)00235-1
(1996)
Cleavage of titanium dimethylamides with methyl iodide

Doi:10.1021/om00019a057
(1994)
Studies on the standardization of crude drugs. XIX. The constituents of Picrasma ailanthoides. I. The structure of nigakinone

Doi:10.1248/yakushi1947.87.11_1371
(1967)
Unusual acetylation of 2-methyl-1-phenylsulfonylindole

Doi:10.1080/00397919608004636
(1996)
α-Diimine-Niobium Complex-Catalyzed Deoxychlorination of Benzyl Ethers with Silicon Tetrachloride

Doi:10.1021/acs.inorgchem.9b01784
(2019)

Article Doi