Synthesis and evaluation of a polyamine phosphinate and phosphonamidate as transition-state analogue inhibitors of spermidine/spermine-N1-acetyltransferase

DOI: 10.1016/0968-0896(96)00072-7

Source and publish data:

Bioorganic and Medicinal Chemistry p. 825 - 836 (1996)

Update date:2022-08-03

Topics:

Authors:

Wu, Ronghui

Saab, Nada H.

Huang, Huatao

Wiest, Laurie

Pegg, Anthony E.

Casero Jr., Robert A.

Woster, Patrick M.

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/0968-0896(96)00072-7

Polyamine analogues such as bis(ethyl)norspermine and N¹-ethyl-N¹¹-[(cyclopropyl)methyl]-4,8-diazaundecane (CPENSpm) act as inhibitors of the enzyme spermidine/spermine-N¹-acetyltransferase (SSAT) in vitro and possess impr

Full text of DOI:10.1016/0968-0896(96)00072-7

Products guided by the article

Product name:1-{N-[benzyloxy(methyl)phosphinyl]amino}-3-[(N,N-dimethyl)amino]propane

Cas No:180523-55-1

R&D Labs maybe for 180523-55-1

Wuhan Yitongtai Science and Technology Co.,Ltd.

Contact:+86-27-88933550

Address:27th Fl. Bldg. 1, Shuian International Mansion, Heping Ave, Wuhan, Hubei, China
JinTan Pingsheng Chemical Co.,Ltd

Contact:+86-519-82828200

Address:NO.11Danfengxilu Road,Jintan City,Jiangsu,China
Hongyi Import & Export CO.,LTD

Contact:86-13319649499

Address:Nanzheng Neighborhood Commitees, Chongwen Office, Yongding District
Shanghai Pengkai Chemical Co.,Ltd

Contact:+86-21-60526671

Address:No.4226 Duzhuang Rd Minhang District Shanghai China
Jiangsu Feymer Technology Co., Ltd.

Contact:+86-512-58110132

Address:Fenghuang Town, Zhangjiagang City, Jiangsu Province, China

Relevant to this article

Synthesis of the D-3 series of phosphatidylinositol phosphates

Doi:10.1021/jo960602u
(1996)
Chemical approaches to bacterial vaccines. Synthesis of mycobacterial oligosaccharide-protein conjugates for use as serodiagnostics and immunogens

Doi:10.1016/0960-894X(96)00235-1
(1996)
Cleavage of titanium dimethylamides with methyl iodide

Doi:10.1021/om00019a057
(1994)
Studies on the standardization of crude drugs. XIX. The constituents of Picrasma ailanthoides. I. The structure of nigakinone

Doi:10.1248/yakushi1947.87.11_1371
(1967)
Unusual acetylation of 2-methyl-1-phenylsulfonylindole

Doi:10.1080/00397919608004636
(1996)
α-Diimine-Niobium Complex-Catalyzed Deoxychlorination of Benzyl Ethers with Silicon Tetrachloride

Doi:10.1021/acs.inorgchem.9b01784
(2019)

Article Doi