
Tetrahedron p. 305 - 318 (1996)
Update date:2022-07-29
Schirlin
Baltzer
Altenburger
Tarnus
Remy
The synthesis of difluoromethyleneketone retroamides is described. Several examples of application to aspartyl or seryl proteases illustrate the versatility of this inactivation concept. Copyright
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