Bioorganic and Medicinal Chemistry Letters p. 2921 - 2926 (1999)
Update date:2022-08-05
Topics:
Jimonet, Patrick
Boireau, Alain
Cheve, Michel
Damour, Dominique
Genevois-Borella, Arielle
Imperato, Assunta
Pratt, Jeremy
Randle, John C. R.
Ribeill, Yves
Stutzmann, Jean-Marie
Mignani, Serge
Original spiro-imidazo[1,2-a]indeno[1,2-e]pyrazine-4-one derivatives were synthesised and led to the identification of 3e which showed good affinities for both the AMPA and the NMDA glycine-site receptors, and displayed good anticonvulsant effects after i
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