Design and Combinatorial Development of Shield-1 Peptide Mimetics Binding to Destabilized FKBP12

DOI: 10.1021/acscombsci.9b00197

Source and publish data:

ACS Combinatorial Science (2020)

Update date:2022-08-02

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Authors:

Bols, Mikael

Diness, Frederik

J?rgensen, Frederik P.

Madsen, Daniel

Meldal, Morten

Olsen, Jakob V.

Palmer, Daniel

Roux, Milena E.

Schoffelen, Sanne

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Article abstract of DOI:10.1021/acscombsci.9b00197

On the basis of computational design, a focused one-bead one-compound library has been prepared on microparticle-encoded PEGA₁₉₀₀ beads consisting of small tripeptides with a triazole-capped N-terminal. The library was screened towards a double

Full text of DOI:10.1021/acscombsci.9b00197

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