Synthesis and highly diastereoselective alkylation of chiral N-[(S,S)-3,5-bis(1-methoxyethyl)-1,2,4-triazol-4-yl]arylimines

DOI: 10.1016/0957-4166(96)00196-6

Source and publish data:

Tetrahedron Asymmetry p. 1621 - 1630 (1996)

Update date:2022-08-02

Topics:

Authors:

Katritzky, Alan R.

El-Zemity, Saad R.

Leeming, Peter

Hartshorn, Chris M.

Steel, Peter J.

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/0957-4166(96)00196-6

(S,S)-4-Amino-3,5-bis(1-hydroxyethyl)-1,2,4-triazole 2 (SAT) (from (S)-lactic acid and hydrazine hydrate) reacted with substituted benzaldehydes 6 to afford N-[(S,S)-3,5-bis(1-hydroxyethyl)-1,2,4-triazol-4-yl]arylimines 3 in excellent yield. Protection of

Full text of DOI:10.1016/0957-4166(96)00196-6

Products guided by the article

Product name:(S)-1-[4-{[1-(4-Chloro-phenyl)-meth-(E)-ylidene]-amino}-5-((S)-1-hydroxy-ethyl)-4H-[1,2,4]triazol-3-yl]-ethanol

Cas No:180857-96-9

R&D Labs maybe for 180857-96-9

uni source industries limited

Contact:86 21 3772 9386

Address:Rm.1803,Starry Bldg.1,1505 Meijiabang Road,Shanghai 201620 China
NOVASYNCS CO., LTD

Contact:0512-63006287

Address:no.88.YISHENG Road,etdz-WUJIANG,SUZHOU,CHINA
Tomo Pharma Chem Co., Limited

Contact:+86-158-05817090

Address:ROOM 9F, FLAT 2, GUODU DEVELOPING BLDG, No.182, ZHAOHUI ROAD
Hebei DaPeng Pharm & Chem Co., Ltd.

Contact:86-317-7298678,0576-88861898 88861908

Address:West Songmen Village, East Songmen Town, Wuqiao, Cangzhou, Hebei ,China
Nanjing Samwon International Limited

Contact:+86-25-84873444

Address:1108, BLDG B, New Century Plaza, No 1, South Taiping Rd.,

Relevant to this article

An unequivocal synthesis of 4-amino-1,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-2,7-diones and 2-amino-3,5,6,8-tetrahydropyrido[2,3-d]pyrimidine-4,7-diones

Doi:10.1135/cccc19960901
(1996)
Biomimetic cyclization of enamide-containing polyenes as a new route to azapolycycles

Doi:10.1021/jo960924y
(1996)
4-[5-Methyl-3-phenylisoxazol-4-yl]-benzenesulfonamide, Valdecoxib: A potent and selective inhibitor of COX-2 [4]

Doi:10.1021/jm990577v
(2000)
Copper-mediated regio- and enantio-selective cross-coupling of heterocyclic allyl sulphides with organomagnesium compounds: A case of 1,7-relative stereogenesis

Doi:10.1016/0040-4020(96)00601-1
(1996)
Molar scale synthesis of enantiopure stilbene oxide

Doi:10.1021/jo960718q
(1996)
Highly effective procedure for introduction of amino group into the 2-position of imidazole ring

Doi:10.3987/com-96-7475
(1996)

Article Doi